small molecule

IMBRUVICA

IBRUTINIB

Loss of exclusivitySeptember 2036latest FDA-listed patent expiry
CompanyPharmacyclicsView the full company profile on CliffBio

Drug detail

Brand nameIMBRUVICA
Active ingredientIBRUTINIB
Strength280MG
Dosage formTABLET
RouteORAL
ModalitySmall molecule
FDA approvalFebruary 2018
Marketing statusRX

Listed patents

PatentExpiresType
9655857*PEDSeptember 2036
10010507*PEDSeptember 2036
10213386*PEDSeptember 2036
10828259*PEDSeptember 2036
10828259March 2036product
12551448March 2036product
10010507March 2036product
10213386March 2036product
9655857March 2036product
10463668*PEDApril 2035
9795604*PEDApril 2035
10695350*PEDApril 2035
10695350October 2034use U-2846
9795604October 2034use U-2970
10463668October 2034use U-2654
9296753*PEDApril 2034
10106548*PEDDecember 2033
10961251*PEDDecember 2033
9725455*PEDDecember 2033
10125140*PEDDecember 2033
9296753October 2033substance
10961251June 2033product
10106548June 2033substance, product
10125140June 2033substance, product
9725455June 2033substance
10004746*PEDDecember 2031
9125889*PEDDecember 2031
9801883*PEDDecember 2031
10016435*PEDDecember 2031
10478439*PEDDecember 2031
8999999*PEDDecember 2031
9801881*PEDDecember 2031
10751342*PEDDecember 2031
11672803June 2031use U-2242
9801883June 2031use U-2159
9125889June 2031use U-1650
8999999June 2031use U-1491
9801881June 2031use U-2242
10004746June 2031use U-2242
10016435June 2031use U-1650
10478439June 2031use U-3422
10751342June 2031use U-1491
8008309*PEDMay 2028
8008309November 2027substance, product
8563563*PEDOctober 2027
8754091*PEDJune 2027
8952015*PEDJune 2027
7514444*PEDJune 2027
8476284*PEDJune 2027
8957079*PEDJune 2027
8703780*PEDJune 2027
8735403*PEDJune 2027
8497277*PEDJune 2027
9181257*PEDJune 2027
8697711*PEDJune 2027
8563563April 2027use U-2241
8703780December 2026use U-1491
8697711December 2026substance, product
9181257December 2026substance
8735403December 2026substance, product
7514444December 2026substance, product
8957079December 2026substance, product
8754091December 2026product
8497277December 2026use U-3422
8476284December 2026use U-1946
8952015December 2026use U-1491

Regulatory exclusivity

CodeExpires
PEDFebruary 2030
ODE-405August 2029
PEDFebruary 2026
NPPAugust 2025

Source: FDA Orange Book, layered on the CliffBio company graph. Cliff dates are the latest FDA-listed patent expiry; estimates are projections, not legal advice.

IMBRUVICA patent cliff — loss of exclusivity September 2036 | CliffBio