small molecule

LUTATHERA

LUTETIUM LU 177 DOTATATE

Loss of exclusivityJanuary 2039latest FDA-listed patent expiry
CompanyADVANCED ACCELERATOR APPLICATIONS USA INC

Drug detail

Brand nameLUTATHERA
Active ingredientLUTETIUM LU 177 DOTATATE
Strength10mCi/ML
Dosage formSOLUTION
RouteINTRAVENOUS
ModalitySmall molecule
FDA approvalJanuary 2018
Marketing statusRX

Listed patents

PatentExpiresType
12168063*PEDJanuary 2039
12415003*PEDJanuary 2039
12144873*PEDJanuary 2039
12151003*PEDJanuary 2039
12491272*PEDJanuary 2039
10596278*PEDJanuary 2039
10596276*PEDJanuary 2039
12161732*PEDJanuary 2039
11904027*PEDJanuary 2039
12168063July 2038product
12415003July 2038use U-4036
12491272July 2038use U-4036
12144873July 2038use U-4036
12151003July 2038product
12161732July 2038product
10596278July 2038product
10596276July 2038product
11904027July 2038product

Regulatory exclusivity

CodeExpires
PEDOctober 2031
ODE-479April 2031
PEDOctober 2027
NPPApril 2027

Source: FDA Orange Book, layered on the CliffBio company graph. Cliff dates are the latest FDA-listed patent expiry; estimates are projections, not legal advice.

LUTATHERA patent cliff — loss of exclusivity January 2039 | CliffBio