small molecule

ORLADEYO

BEROTRALSTAT DIHYDROCHLORIDE

Loss of exclusivityMay 2040latest FDA-listed patent expiry
CompanyBioCryst PharmaceuticalsView the full company profile on CliffBio

Drug detail

Brand nameORLADEYO
Active ingredientBEROTRALSTAT DIHYDROCHLORIDE
StrengthEQ 150MG BASE
Dosage formCAPSULE
RouteORAL
ModalitySmall molecule
FDA approvalDecember 2020
Marketing statusRX

Listed patents

PatentExpiresType
12545646*PEDMay 2040
11117867*PEDMay 2040
12545647*PEDMay 2040
10662160*PEDMay 2040
12552750*PEDMay 2040
12545645*PEDMay 2040
12344585*PEDMay 2040
11618733*PEDMay 2040
12590069*PEDMay 2040
12590068*PEDMay 2040
11117867November 2039product
12344585November 2039use U-3010
10662160November 2039substance
11618733November 2039use U-3300
12545646November 2039substance, product
12590068November 2039substance, product
12590069November 2039substance, product
12545647November 2039substance, product
12545645November 2039substance, product
12552750November 2039substance, product
10125102*PEDOctober 2035
11708333*PEDSeptember 2035
12116346*PEDSeptember 2035
11230530*PEDSeptember 2035
10689346*PEDSeptember 2035
10329260*PEDSeptember 2035
10125102April 2035substance
11708333March 2035use U-3300
10329260March 2035substance
11230530March 2035use U-3300
12116346March 2035substance
10689346March 2035use U-3010

Regulatory exclusivity

CodeExpires
PEDJune 2028
ODE-333December 2027

Source: FDA Orange Book, layered on the CliffBio company graph. Cliff dates are the latest FDA-listed patent expiry; estimates are projections, not legal advice.

ORLADEYO patent cliff — loss of exclusivity May 2040 | CliffBio