small molecule

AKYNZEO

FOSNETUPITANT CHLORIDE HYDROCHLORIDE; PALONOSETRON HYDROCHLORIDE

Loss of exclusivityJune 2037latest FDA-listed patent expiry
CompanyHELSINN HEALTHCARE SA

Drug detail

Brand nameAKYNZEO
Active ingredientFOSNETUPITANT CHLORIDE HYDROCHLORIDE; PALONOSETRON HYDROCHLORIDE
StrengthEQ 235MG BASE/20ML (EQ 11.75MG BASE/ML);EQ 0.25MG BASE/20ML (EQ 0.0125MG BASE/ML)
Dosage formSOLUTION
RouteINTRAVENOUS
ModalitySmall molecule
FDA approvalMay 2020
Marketing statusRX

Listed patents

PatentExpiresType
11529362June 2037product
10624911June 2037product
12208109June 2037product
11312698May 2032substance, product
9908907May 2032substance, product
8426450May 2032substance, product
10717721May 2032substance
9403772May 2032substance
10208073May 2032use U-2301
8895586May 2032use U-2301
10828297December 2030use U-2301
9186357November 2030use U-2301

Source: FDA Orange Book, layered on the CliffBio company graph. Cliff dates are the latest FDA-listed patent expiry; estimates are projections, not legal advice.