small molecule

KALYDECO

IVACAFTOR

Loss of exclusivityAugust 2033latest FDA-listed patent expiry
CompanyVERTEX PHARMACEUTICALS INC

Drug detail

Brand nameKALYDECO
Active ingredientIVACAFTOR
Strength13.4MG/PACKET
Dosage formGRANULE
RouteORAL
ModalitySmall molecule
FDA approvalMay 2023
Marketing statusRX

Listed patents

PatentExpiresType
10272046*PEDAugust 2033
11752106*PEDAugust 2033
12214083*PEDAugust 2033
11147770*PEDAugust 2033
8883206*PEDAugust 2033
8883206February 2033product
11147770February 2033product
12214083February 2033product
11752106February 2033product
10272046February 2033product
12458635*PEDFebruary 2030
11564916*PEDFebruary 2030
10646481*PEDFebruary 2030
11564916August 2029use U-3603
12458635August 2029product
10646481August 2029product
8324242*PEDFebruary 2028
7495103*PEDNovember 2027
8324242August 2027use U-3609
8754224*PEDJune 2027
9670163*PEDJune 2027
8410274*PEDJune 2027
7495103May 2027substance, product
8354427*PEDJanuary 2027
8754224December 2026substance, product
9670163December 2026product
8410274December 2026product
8354427July 2026use U-3608

Regulatory exclusivity

CodeExpires
PEDNovember 2030
ODE-435May 2030
PEDNovember 2028
M-14May 2028
PEDNovember 2026
NPPMay 2026

Source: FDA Orange Book, layered on the CliffBio company graph. Cliff dates are the latest FDA-listed patent expiry; estimates are projections, not legal advice.

KALYDECO patent cliff — loss of exclusivity August 2033 | CliffBio